平安! 发表于 2011-11-9 19:57 4 ^! v1 x7 J& F
Pazopanib (100 mg/kg/day free base equivalent)
+ \9 A; S. ?. P' x 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。% [# g( l, A) P
搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。8 k Y; k5 o$ }4 u$ u
7 K" S: w1 Z) r( a# w* ?以下是正版说明书的推荐用量。
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--------------------- DOSAGE AND ADMINISTRATION ----------------
# d; J6 O! Q% l8 e9 i* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) % W: K" H1 Y* f% Y4 W* }
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
/ R" h' P9 Z Y( ?1 z, E) u$ D+ A---------------------DOSAGE FORMS AND STRENGTHS --------------
, ^7 G1 ?' d& E2 ?200 mg tablets. (3) " Q$ q( C s, k2 i( R# M' X
-------------------------------CONTRAINDICATIONS------------------------ |